De Novo Design of a Picomolar Nonbasic 5-HT1B Receptor Antagonist

Nugiel, D.A.; Krumrine, J.R.; Hill, D.C.; Damewood, J.R.; Bernstein, P.R.; Sobotka-Briner, C.D.; Liu, J.W.; Zacco, A.; Pierson, M.E.; De Novo Design of a Picomolar Nonbasic 5-HT1B Receptor Antagonist; J. Med. Chem.; 2010; 53; 1876-1880
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